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Diroximel Fumarete

CAS No. 1577222-14-0

Diroximel Fumarete ( Diroximel fumarate; ALKS8700; ALKS 8700; ALKS-8700 )

产品货号. M17336 CAS No. 1577222-14-0

Diroximel fumarate, a prodrug of monomethyl fumarate in a controlled-release formulation, rapidly and potently converts to MMF in the body.

纯度: 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥429 有现货
5MG ¥721 有现货
10MG ¥1037 有现货
25MG ¥1823 有现货
50MG ¥2811 有现货
100MG ¥4528 有现货
500MG ¥9639 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Diroximel Fumarete
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Diroximel fumarate, a prodrug of monomethyl fumarate in a controlled-release formulation, rapidly and potently converts to MMF in the body.
  • 产品描述
    Diroximel fumarate, also known as ALKS-8700, is a prodrug of monomethyl fumarate in a controlled-release formulation that rapidly and efficiently converts to MMF in the body.
  • 同义词
    Diroximel fumarate; ALKS8700; ALKS 8700; ALKS-8700
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    Others
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1577222-14-0
  • 分子量
    255.22
  • 分子式
    C11H13NO6
  • 纯度
    98%
  • 溶解度
    DMSO : 125 mg/mL. 489.77 mM;
  • SMILES
    COC(=O)/C=C/C(=O)OCCN1C(=O)CCC1=O
  • 化学全称
    2-(2,5-dioxopyrrolidin-1-yl)ethyl methyl fumarate

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Alkermes Announces Positive Clinical Trial Results and Streamlined Registration Pathway for ALKS 8700 for Treatment of Multiple Sclerosis. October 29, 2015 07:00 AM Eastern Daylight Time.
产品手册
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